| Year | Name | Institution |
|---|---|---|
| 1978 | Tadao Uyehara | Tohoku University, Japan |
| 1984 | John Steven Taylor | Washington University, St. Louis |
| 1985 | Tadhg Begley | Texas A&M |
| 1985 | Peter G. Schultz | The Scripps Research Institute |
| 1988 | Michael Van Dyke | Kennesaw State University |
| 1989 | Alanna Schepartz | Yale University |
| 1989 | Sam Gellman | University of Wisconsin, Madison |
| 1990 | James E. Hanson | Seton Hall University |
| 1990 | Paul Kamer | University of Amsterdam |
| 1990 | John Termini | City of Hope |
| 1990 | Eric Kool | Stanford University |
| 1990 | Marc M. Greenberg | Johns Hopkins University |
| 1990 | Brent Iverson | University of Texas, Austin |
| 1991 | L. J. I. Maher III | Mayo Foundation, Rochester, MN |
| 1991 | David Horne | City of Hope |
| 1991 | Laura Kiessling | Massachusetts Institute of Technology |
| 1992 | Kent Gates | University of Missouri |
| 1992 | Mark Distefano | University of Minnesota |
| 1992 | Erick Carreira | ETH-Zürich, Switzerland |
| 1993 | Yitzhak Tor | University of California, San Diego |
| 1994 | Jumi Shin | University of Toronto |
| 1994 | Ken Turnbull | University of Arkansas |
| 1994 | Stephen Woski | University of Alabama |
| 1995 | Scott Strobel | Yale University |
| 1996 | Jürg Hunziker | Universität Bern, Switzerland |
| 1996 | Martha Oakley | Indiana University |
| 1996 | Milan Mrksich | Northwestern University |
| 1996 | Peter Beal | University of California, Davis |
| 1996 | Scott Singleton | University of North Carolina |
| 1996 | Jon Parquette | Ohio State University |
| 1997 | Robert H. E. Hudson | University of Western Ontario |
| 1997 | Kathy B. Grant | Georgia State University |
| 1998 | Hogyu Han | Korea University, Seoul |
| 1999 | David Liberles | Temple University |
| 1999 | Paul Floreancig | University of Pittsburgh |
| 1999 | Simon Friedman | University of Missouri, Kansas City |
| 2000 | Joseph Hacia | University of Southern California Keck School of Medicine |
| 2000 | Ulf Ellervik | Lund University, Sweden |
| 2000 | Anna K. Mapp | University of Michigan |
| 2000 | Robert Haner | University of Bern, Switzerland |
| 2000 | Kevin Luebke | University of Texas Southwestern Medical Center |
| 2001 | Thomas Minehan | Cal State University, Northridge |
| 2002 | Paramjit (Bobby) Arora | New York University |
| 2003 | Z. Y. (James) Zhan | Fudan University, Shanghai |
| 2003 | Alexander Heckel | Goethe Universitat, Frankfurt am Main |
| 2003 | Clay C. C. Wang | University of Southern California School of Pharmacy |
| 2004 | Leonard J. Prins | University of Padova, Italy |
| 2004 | Adam R. Urbach | Trinity University |
| 2004 | Christian Melander | North Carolina State University |
| 2004 | Hans-Dieter Arndt | Max-Planck Institute, Dortmund |
| 2005 | Jason Belitsky | Oberlin College |
| 2006 | Shane Foister | University of Tennessee |
| 2009 | Daniel Harki | University of Minnesota-Twin Cities |
| 2010 | David Chenoweth | University of Pennsylvania |
| 2013 | Amanda Hargrove | Duke University |
| 2013 | Chieh-Mei (Jamie) Wang | West China College, Sichuan University |
| 2013 | Michelle Farkas | University of Massachusetts Amherst |
| 2014 | Jevgenij Raskatov | University of California, Santa Cruz |
| 2014 | Nicholas Nickols | UCLA Medical School |
| 2014 | Zhiwei Yang | Beijing College of Chemical Technology |
| 2015 | Amanda Silberstein | Westmont College |
| 2015 | Alissa Hare | Vanderbilt University |
| 2017 | Karen Draths | Michigan State University |
| 2018 | Tiezheng Jia | SUSTech, Shenzhen |
| 2020 | Jerzy Szablowski | Rice University |
| 2021 | Thomas Martinez | UC Irvine |